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Valproate

Composition

Contains Valproic acid or its derivatives, an anticonvulsant and mood stabilizer.

Indications

Used to treat epilepsy, bipolar disorder , and migraine prophylaxis.

Side effects

Weight gain, tremor, drowsiness, hair loss, GI upset, liver toxicity, thrombocytopenia.

Precautions

Monitor liver function and platelets; use with caution in pregnancy due to teratogenicity

Contraindications

Liver disease, known urea cycle disorders, mitochondrial disorders , pregnancy.

Dosage and administration

Individualized dosing; commonly 10–60 mg/kg/day in divided doses.

Countries

Mexico, Brazil, Colombia

Available Forms

Oral tablets (immediate and extended-release), capsules, syrup, and injectable formulations.